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The Smelly Way
April 1, 2010
· New Papers

From Carboxylic Acids to the Trifluoromethyl Group Using BrF3 A method to convert carboxylic acids into trifluoromethyl groups. This paper by…

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From Boronic Acids to Aminoacids
April 1, 2010
· New Papers

Synthesis of Unnatural Amino Acid Derivatives via Palladium-catalyzed 1,4-Addition of Boronic Acids Take advantage of many boronic acids to get unnatural…

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Back in the Chain Gang
April 1, 2010
· New Papers

Direct Synthesis of Cbz-protected (2-Amino)-6-(2-aminoethyl)pyridines Construction of ethylamino chains over functionalized pyridines and other azoles. The importance of the 2-amino-6-(2-aminoethyl)pyridine skeleton…

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Optimum Ratio
April 1, 2010
· New Papers

Mild and General Method for the a-Arylation of Heteroaromatic Ketones With heterocycles, sometimes it is worth to check the ligand to…

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One Thousand and One Nights
April 1, 2010
· New Papers

Triethanolamine-Mediated Palladium-Catalyzed Regioselective C-2 Direct Arylation of Free NH-Pyrroles Arylation of pyrroles using a phosphine-free protocol. ‘C-H activation is one of…

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A Nickel For a Ketone
April 1, 2010
· New Papers

Direct Synthesis of Arylketones by Nickel-Catalyzed Addition of Arylboronic Acids to Nitriles Ketones from boronic acids and nitriles One of the…

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Not Only with Triflates
April 1, 2010
· New Papers

Pd-Catalyzed Cross-Coupling Reactions of Amides and Aryl Mesylates Still thinking about triflates for a coupling? Think again. The introduction of a…

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Titanium Is the Key
April 1, 2010
· New Papers

Titanium(IV) Isopropoxide Mediated Synthesis of Pyrimidin-4-ones Synthesis of highly substituted pyrimidones from amides mediated by Titanium. The pyrimidin-4-one scaffold is widespread…

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More C-H activation
April 1, 2010
· New Papers

Copper-Catalyzed Amination of Primary Benzylic C-H Bonds with Primary and Secondary Sulfonamides Once again a case of C-H activation, this time…

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Very Ir-teresting
April 1, 2010
· New Papers

Iridium-Catalyzed a-Alkylation of Acetates with Primary Alcohols and Diols A method for the alkylation of acetates using Iridium. Aldolic condensation is…

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